Synthesis of pterocellin A.
نویسندگان
چکیده
The first total synthesis of pterocellin A (1) was achieved in 10 linear steps from commercially available kojic acid (6) and 2-bromo-3-pyridinol (11) in a convergent sequence. The key constructive steps are a directed lithiation to couple two pyridines and an intramolecular nucleophilic aromatic substitution to form 1. [structure: see text]
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ورودعنوان ژورنال:
- Organic letters
دوره 8 12 شماره
صفحات -
تاریخ انتشار 2006